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    • Dr. Meckler's U.S. Patents:

    1. Popp, K.; Meckler, H. Methods of Treatment using Amphetamine Controlled Release, Prodrug and Abuse Resistant Dosage Forms. U.S. Patent 11,717,498; August 8, 2023.

    2. Popp et al. Amphetamine Controlled Release, Prodrug, and Abuse-Deterrent Dosage Forms. U.S. Patent 11,123,310; September 21, 2021.

    3. Meckler, H.; Gregg, B.T.; Yang, J. Chiral Aziridine Phosphoramidate Compounds. U.S. Patent 10,087,202; October 2, 2018.

    4. Meckler, H.; Gregg, B.T.; Yang, J. Novel Chiral Aryl or Aryl-Alkyl Phosphoramidate Dexamphetamine Precursors Having A Regioisomeric Purity >99%. U.S. Patent 9,657,041; May 23, 2017.

    5. Meckler, H.; Gregg, B.T.; Yang, J. Synthesis of Racemic Amphetamine Derivatives by Cuprate Addition Reaction with Aziridine Phosphoramidate Compounds. U.S. Patent 9,321,794; April 26, 2016.

    6. Meckler, H.; Gregg, B.T.; Yang, J. Synthesis of Chiral Amphetamine Derivatives by Stereospecific, Regioselective Cuprate Addition Reaction with Aziridine Phosphoramidate Compounds. U.S. Patent 9,278,904; March 8, 2016.

    7. Boulanger, W.A.; Collier, S.J.; Eastham, S.A.; Edie, D.L.; Guevel, R.Y.; Hernandez-Abad, P.E.; Herr, J.R.; Kjaersgaard, H.J.; Meckler, H.; Polomski, R.E.; Schow, S.R.; Zhichkin, P. E. U.S. Process for and intermediates in the preparation of canfosfamide and its salts. U.S. Patent. 8,334,266, Dec. 18, 2012.

    8. Boulanger, W.A.; Edie, D.L.; Guevel, R.Y.; Hernandez-Abad, P.E.; Herr, J.R.; Meckler, H.; Schow, S.R.; Zhichkin, P. E. U.S. Process for and intermediates in the preparation of canfosfamide and its salts. U.S. Patent. 8,198,247, June 12, 2012.

    9. Burdick, D.C.; Collier, S. J.; Biolatto, B.; Meckler, H. Process for production of delta-9-tetrahydrocannabinol. U.S. Patent 8,106,244, January 31, 2012.

    10. Meckler, H.; Littler, B.; Raje, P.; Van Brunt, M.; Vogt, P.F. Process for production of Piperidine derivatives. U.S. Patent 8,067,605, November 29, 2011.

    11. Meckler, H.; Littler, B.; Raje, P.; Van Brunt, M.; Vogt, P.F. Process for production of carebastine. U.S. Patent 8,067,604, November 29, 2011.

    12. Meckler, H.; Littler, B. J.; Raje, P.; Van Brunt, M.; Vogt, P. F. Process for Production of Piperidine Derivatives. U.S. Patent 7,863,452, January 4, 2011.

    13. Meckler, H.; Littler, B. J.; Raje, P.; Van Brunt, M.; Vogt, P. F. Process for Production of Carebastine. U.S. Patent 7,858,798, December 28, 2010.

    14. Burdick, D. C.; Collier, S. J.; Jos, F.; Biolatto, B.; Paul, B. J.; Meckler, H.; Helle, M. A.; Habershaw, A. J. Process for production of delta-9-tetrahydrocannabinol. U.S. Patent 7,674,922. March 9, 2010.

    15. Meckler, H.; Littler, B. J.; Raje, P.; Van Brunt, M.; Vogt, P. F. Process for production of carebastine. U.S. Patent 7,498,443, March 3, 2009.

    16. Meckler, H.; Littler, B.; Raje, P.; Van Brunt, M.; Vogt, P. F. Process for production of piperidine derivatives. U.S. Patent 7,498,345, March 3, 2009.

    17. Kinney, W. A.; Jones, S.; Zhang, X.; Rao, M. N.; Bulliard, M.; Meckler, H.; Lee, N. Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds U.S. Patent 6,610,866, August 26, 2003.

    18. Meckler, H.; Helle, M. A.; Geiss, W. B.; Gregg, B. T. Stereoselective preparation of 24(S)-hydroxyvitamin D2 via coupling reaction U.S. Patent 6,359,012, March 19, 2002.

    19. Kinney, W. A.; Jones, S.; Zhang, X.; Rao, M. N.; Bulliard, M.; Meckler, H.; Lee, N. Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds U.S. Patent 6,262,283, July 17, 2001.

    20. Scott, I. L.; Kogan, T. P.; Meckler, H. Preparation and stereoselective glucosidation of tetra-O-pivaloylmannopyranosyl fluoride U.S. Patent 5,712,387, January 27, 1998.

    21. Wasley, J. W. F.; Gelotte, K. O.; Meckler, H. Preparation and formulation of (pyrrolophenyl)alkanamides and analogs as lipoxygenase inhibitors U.S. Patent 5,096,919, March 17, 1992.

    Dr. Meckler's International Patents:

    1. Meckler, H.; Cleary, D.; Brackeen, M.; Suryadevara, P. Process for Making Levoamphetamine. UK Patent GB2595995; September 13, 2023.

    2. Popp et al. Amphetamine Controlled Release, Prodrug, and Abuse-Deterrent Dosage Forms. Israeli Patent 261,366; June 2, 2022.